Official Title
Imaging of Patients With Solid Tumor Cancer Via Intermediate-Size Patient Population Expanded Access Investigational New Drug (IND)
Brief Summary

The purpose of this Expanded Access Program (EAP) is to allow use of the investigationalimaging agent, MNPR-101-DFO*-89Zr, with positron emission tomography/computed tomography(PET/CT) imaging, to non-invasively detect the presence of urokinase plasminogenactivator receptor (uPAR) binding in solid tumors. uPAR binding is higher in tumorscompared to normal tissue in some cancers.

Detailed Description

Imaging agent MNPR-101-DFO*-89Zr will be dosed to adult patients diagnosed with solid
tumor cancer followed 3 to 5 days later by PET/CT imaging. The result will determine if
there is sufficient uPAR binding, as assessed by the Investigator, to support
administration of the companion intervention MNPR-101-PCTA-177Lu in a separate expanded
access program (EAP IST-00Cb). The safety of MNPR-101-DFO*-89Zr will be evaluated as will
the amount of radioactivity present in blood samples.

Available
Intermediate-size Population
Cancer
Solid Tumor
Solid Tumor, Adult

Diagnostic Test: MNPR-101-DFO*-89Zr

MNPR-101-DFO*-89Zr is an antibody radionuclide conjugate intended to image solid tumors
expressing uPAR.

Eligibility Criteria

Key Inclusion Criteria:

- Histologically or cytologically confirmed locally advanced or metastatic solid tumor
cancer that is refractory to existing therapy(ies) known to provide clinical
benefit, or for which no standard treatment is available, or is contraindicated

- Ability to understand and willingness to sign a written informed consent document

Key Exclusion Criteria:

- Continuing ≥ Grade 3 adverse reactions from prior systemic therapy (Common
Terminology Criteria for Adverse Events [CTCAE] version 5.0)

- Prior treatment with any radiopharmaceutical or investigational agents within 4
weeks or 5 half-lives, whichever is longer, prior to administration of
MNPR-101-DFO*-89Zr

- Evidence of impaired organ function, particularly bone marrow, liver, kidney, or
heart, according to specific test parameters

- Presence of other serious, non-malignant diseases or any other condition that, in
the opinion of the investigator, could interfere with the objectives of the study,
participant safety, or compliance.

Eligibility Gender
All
Eligibility Age
Minimum: 18 Years ~ Maximum: N/A
Countries
United States
Locations

Excel Diagnostics & Nuclear Oncology Center
Houston, Texas, United States

Contacts

Susan Cork, Therapy Coordinator
+1 713-781-6200 - Ext. 3203
scork@exceldiagnostics.com

Nereyda Sauceda, Therapy Coordinator
+1 713-781-6200 - Ext. 3246
nsauceda@exceldiagnostics.com

Ebrahim S. Delpassand, M.D. Chairman & Medical Director, Nuclear Medicine, Principal Investigator
Excel Diagnostics & Nuclear Oncology Center

Monopar Therapeutics
NCT Number
Keywords
Solid tumor
PET/CT
urokinase plasminogen activator receptor
uPAR
Zirconium-89 imaging
Positron emission tomography/computed tomography
MNPR-101-DFO*-89Zr
uPAR-positive
Urokinase plasminogen activator receptor-positive
EAP IST-00Cb
Antibody radionuclide conjugate
Monoclonal antibody radionuclide conjugate
Solid tumor imaging
MeSH Terms
Neoplasms