Official Title
A Phase 3, Randomized, Placebo-Controlled, Double-Blind Clinical Study to Evaluate the Efficacy and Safety of Molnupiravir (MK-4482) in Non-Hospitalized Adults With COVID-19 at High Risk for Disease Progression
Brief Summary

Researchers are looking for other ways to prevent severe illness from COVID-19. COVID-19is a virus that most often causes mild flu or cold-like symptoms. However, people withcertain health conditions or other factors have a high risk (chance) of getting severelyill from COVID-19, which can require a hospital stay or lead to death. Some people whoare high risk for severe illness may be unable to take certain treatments for COVID-19because they are not available to them, or they take other medicines that may react witha treatment and cause an unwanted effect.Molnupiravir (MK-4482) is a study medicine designed to stop the COVID-19 virus fromcopying itself in the body (multiplying). The goal of this study is to learn ifmolnupiravir prevents severe illness from COVID-19 more than placebo in people who arehigh risk.

Detailed Description

Not Provided

Recruiting
Coronavirus Disease (COVID-19)

Drug: Molnupiravir

Molnupiravir administered orally as two 400 mg film-coated tablets every 12 hours for 5
days (a total of 10 consecutive doses)
Other Name: MK-4482,LAGEVRIO®

Drug: Placebo

Molnupiravir-matching placebo administered orally as two film-coated tablets every 12
hours for 5 days (a total of 10 consecutive doses)

Eligibility Criteria

Inclusion Criteria

The main inclusion criteria include but are not limited to the following:

- Is an individual of any sex/gender, ≥18 years of age

- Has documentation of SARS-CoV-2 infection with sample collection ≤4 days prior to
randomization

- Has initial onset of signs/symptoms attributable to COVID-19 for ≤4 days prior to
the day of randomization and ≥2 of the following signs/symptoms attributable to
COVID-19 on the day of randomization: cough, sore throat, nasal congestion,
shortness of breath or difficulty breathing with exertion, muscle or body aches,
fatigue, fever >38.0°C or chills, nausea or vomiting or diarrhea, change in sense of
smell or change in sense of taste, or headache

- Has ≥1 of the following characteristics or medical conditions associated with the
highest risk of severe illness from COVID-19:

- Advanced age of ≥75 years of age

- Immunocompromised

- Neurocognitive or physical disability

- Has ≥3 characteristics or medical conditions which increase the risk of severe
illness due to COVID-19 (e.g., chronic lung disease, obesity with body mass index
≥35, diabetes)

- Is unable to receive treatment with nirmatrelvir/ritonavir (NMV/r) due to 1 or more
of the following:

- Is receiving drug(s) highly dependent on cytochrome P450 3A (CYP3A) for
clearance and for which elevated concentrations are associated with serious
and/or life-threatening consequences or drug(s) with a clinically significant
drug-drug interaction for which co-administration is not possible

- Is receiving potent CYP3A inducers where significantly reduced nirmatrelvir or
ritonavir plasma concentrations may be associated with the potential for loss
of virologic response and possible resistance

- Has severe renal or hepatic impairment

- Has experienced prior adverse reactions or hepatotoxicity to NMV/r that would
preclude future use

- Has uncontrolled HIV infection

- Has known or suspected NMV/r resistance

- NMV/r is not approved/authorized in the participant's country or it is not
accessible to participant (e.g., drug shortage)

Inclusion note: Participants may receive remdesivir as standard of care in addition to
molnupiravir or placebo. If remdesivir is available and clinically appropriate per local
clinical practice, investigators will aim to ensure that those who are most vulnerable to
severe COVID-19 receive timely access to remdesivir as standard of care on this study.

Exclusion Criteria

The main exclusion criteria include but are not limited to the following:

- Is currently hospitalized or is expected to need hospitalization for COVID-19
imminently

- Has received or plans to receive SARS-CoV-2 directed antivirals or monoclonal
antibodies for current episode of COVID-19 (other than study intervention and, if
applicable, remdesivir as standard of care)

- Has ≥1 of the following signs/symptoms that are attributable to severe or critical
COVID-19:

- Shortness of breath at rest

- Respiratory rate ≥30 breaths per minute

- Heart rate ≥125 beats per minute

- Peripheral oxygen saturation (SpO2) ≤93% on room air or on supplemental oxygen
for a reason other than COVID-19 which has not increased since onset of
COVID-19 signs/symptoms

- Is receiving >4 liters/minute supplemental oxygen for COVID-19 (but was not
receiving supplemental oxygen prior to COVID-19), regardless of SpO2

- Has received a COVID-19 vaccine within 30 days prior to randomization

- Has a history of SARS-CoV-2 infection (with or without symptoms) within 30 days
prior to randomization

- Has known or suspected hypersensitivity to active or inactive ingredients of
molnupiravir

Eligibility Gender
All
Eligibility Age
Minimum: 18 Years ~ Maximum: N/A
Countries
Argentina
Bulgaria
Finland
France
Germany
Italy
Japan
Korea, Republic of
New Zealand
Poland
Puerto Rico
Romania
Spain
Taiwan
Ukraine
United Kingdom
United States
Locations

Cullman Clinical Trials ( Site 3813)
Cullman, Alabama, United States

Helios Clinical Research ( Site 3826)
Paradise Valley, Arizona, United States

Absolute Clinical Research ( Site 3709)
Phoenix, Arizona, United States

Clinica de Salud del Valle de Salinas ( Site 3825)
Castroville, California, United States

Ascada Health PC dba Ascada Research ( Site 3750)
Fullerton, California, United States

Pacific Clinical Studies ( Site 3827)
Los Alamitos, California, United States

Valley Clinical Trials, Inc. ( Site 3707)
Northridge, California, United States

FOMAT Medical Research ( Site 3720)
Oxnard, California, United States

Paradigm Clinical Research, LLC ( Site 3785)
San Diego, California, United States

Optimus Medical ( Site 3817)
San Francisco, California, United States

Millennium Clinical Trials ( Site 3758)
Westlake Village, California, United States

Paradigm Clinical Research Centers, Inc ( Site 3718)
Wheat Ridge, Colorado, United States

Encore Medical Research of Boynton Beach ( Site 3701)
Boynton Beach, Florida, United States

Prestige Clinical Research Center ( Site 3722)
Coral Gables, Florida, United States

Indago Research & Health Center, Inc ( Site 3714)
Hialeah, Florida, United States

Prestige Clinical Research ( Site 3830)
Homestead, Florida, United States

Accel Research Sites Network - St. Pete-Largo Clinical Research Unit ( Site 3779)
Largo, Florida, United States

Clinical Site Partners, LLC dba Flourish Research ( Site 3717)
Leesburg, Florida, United States

Advanced Pulmonary Research Institute ( Site 3781)
Loxahatchee Groves, Florida, United States

Palm Springs Community Health Center ( Site 3757)
Miami Lakes, Florida, United States

Panax Clinical Research ( Site 3803)
Miami Lakes, Florida, United States

Southern Clinical Research ( Site 3773)
Miami, Florida, United States

Florida Pharmaceutical Research and Associates ( Site 3763)
Miami, Florida, United States

Bio-Medical Research LLC ( Site 3804)
Miami, Florida, United States

Bright Research Center ( Site 3746)
Miami, Florida, United States

Miami Clinical Research ( Site 3729)
Miami, Florida, United States

Reed Medical Research ( Site 3761)
Miami, Florida, United States

Combined Research Orlando Phase I-IV ( Site 3797)
Orlando, Florida, United States

CDC Research Institute ( Site 3716)
Port Saint Lucie, Florida, United States

New Tampa Health ( Site 3764)
Tampa, Florida, United States

Clinical Research Trials of Florida ( Site 3703)
Tampa, Florida, United States

Precision Research Center ( Site 3704)
Tampa, Florida, United States

Encore Medical Research - Weston ( Site 3708)
Weston, Florida, United States

Balanced Life Health Care Solutions/SKYCRNG ( Site 3713)
Lawrenceville, Georgia, United States

Renew Health Clinical Research ( Site 3760)
Snellville, Georgia, United States

Rophe Adult and Pediatric Medicine/SKYCRNG ( Site 3816)
Union City, Georgia, United States

Paradigm Clinical Research - Boise ( Site 3841)
Boise, Idaho, United States

University of Louisville School of Medicine ( Site 3706)
Louisville, Kentucky, United States

Barnum Medical Research ( Site 3828)
Natchitoches, Louisiana, United States

Annapolis Internal Medicine - CCT Research ( Site 3700)
Annapolis, Maryland, United States

Kur Research - Columbia Medical ( Site 3767)
Columbia, Maryland, United States

Revival Research Institute, LLC ( Site 3835)
Dearborn, Michigan, United States

Michigan Center of Medical Research (MICHMER) ( Site 3734)
Farmington Hills, Michigan, United States

Henry Ford St John TM Center for Infectious Disease Research ( Site 3766)
Grosse Pointe Woods, Michigan, United States

Mankato Clinic ( Site 3842)
Mankato, Minnesota, United States

Prime Health and Wellness/SKYCRNG ( Site 3726)
Fayette, Mississippi, United States

SKY Integrative Medical Center/SKYCRNG ( Site 3740)
Ridgeland, Mississippi, United States

Nevada Health Centers ( Site 3840)
Carson City, Nevada, United States

WR-CRCN, LLC ( Site 3818)
Las Vegas, Nevada, United States

Holy Name Medical Center ( Site 3807)
Teaneck, New Jersey, United States

Prime Global Research ( Site 3731)
Bronx, New York, United States

OnSite Clinical Solutions ( Site 3784)
Charlotte, North Carolina, United States

Monroe Biomedical Research ( Site 3732)
Monroe, North Carolina, United States

IMA Clinical Research Mount Airy ( Site 3745)
Mount Airy, North Carolina, United States

Research Innovations, LLC ( Site 3712)
Beavercreek, Ohio, United States

Midlands Neurology & Pain Associates ( Site 3751)
Columbia, South Carolina, United States

Helios Clinical Research - JAC ( Site 3833)
Jackson, Tennessee, United States

Javara - Privia Medical Group Gulf Coast - The Woodlands HWH ( Site 3837)
Conroe, Texas, United States

South Texas Clinical Research ( Site 3815)
Corpus Christi, Texas, United States

Care United Research, LLC ( Site 3747)
Forney, Texas, United States

Andres Garcia Zuniga, M.D., P.A. ( Site 3782)
Laredo, Texas, United States

LinQ Research ( Site 3824)
Pearland, Texas, United States

Crossroads Clinical Research-Family Practice ( Site 3739)
Victoria, Texas, United States

Eastside Research Associates ( Site 3727)
Redmond, Washington, United States

CEMIC ( Site 0101)
Buenos Aires., Buenos Aires, Argentina

Instituto de Investigaciones Clinicas Mar del Plata ( Site 0111)
Mar del Plata, Buenos Aires, Argentina

Medconsult Pleven - Lovech ( Site 0501)
Lovech, Bulgaria

Medical Center Hera ( Site 0507)
Montana, Bulgaria

Medconsult Pleven ( Site 0503)
Pleven, Bulgaria

DKC V - Plovdiv ( Site 0508)
Plovdiv, Bulgaria

Medical Center Hera EOOD ( Site 0505)
Sofia, Bulgaria

MeVac - Meilahti Vaccine Research Center ( Site 1200)
Helsinki, Uusimaa, Finland

Centre Hospitalier Universitaire Dijon Bourgogne - Hôpital F-Centre d'Investigation Clinique - Plur
Dijon, Bourgogne, France

Pitie Salpetriere University Hospital-Infectious Disease - Tropical Diseases ( Site 1300)
Paris, Ile-de-France, France

CHU de Saint-Etienne ( Site 1302)
Saint Priest en Jarez, Loire, France

centre hospitalier lyon sud ( Site 1303)
Pierre-Bénite, Rhone, France

klinikum rechts der isar der technischen universität münchen ( Site 1502)
Munchen, Bayern, Germany

IRCCS Azienda Ospedaliero-Universitaria di Bologna, Policlinico di Sant'Orsola ( Site 1904)
Bologna, Italy

Ospedale San Martino ( Site 1900)
Genova, Italy

ASST Fatebenefratelli Sacco ( Site 1901)
Milano, Italy

AOU Pisana- Ospedale Cisanello ( Site 1905)
Pisa, Italy

Sekino Hospital ( Site 2016)
Toshimaku, Tokyo, Japan

Wonju Severance Christian Hospital-Internal Medicine ( Site 3009)
Wonju, Kang-won-do, Korea, Republic of

Chonnam National University Hospital-Infectious Diseases ( Site 3008)
Gwangju-si, Kwangju-Kwangyokshi, Korea, Republic of

Korea University Ansan Hospital ( Site 3007)
Ansan-si, Kyonggi-do, Korea, Republic of

Gyeongsang National University Hospital ( Site 3005)
Jinju-si, Kyongsangnam-do, Korea, Republic of

Pusan National University Hospital-Internal Medicine ( Site 3010)
Pusan, Pusan-Kwangyokshi, Korea, Republic of

Kyungpook National University Chilgok Hospital-Division of Infectious Diseases ( Site 3002)
Deagu, Taegu-Kwangyokshi, Korea, Republic of

Korea University Anam Hospital ( Site 3001)
Seoul, Korea, Republic of

Hallym University Kangnam Sacred Heart Hospital-Internal Medicine ( Site 3003)
Seoul, Korea, Republic of

Korea University Guro Hospital ( Site 3006)
Seoul, Korea, Republic of

CGM Research Trust ( Site 2307)
Christchurch, Canterbury, New Zealand

Pacific Clinical Research Network - Tasman ( Site 2304)
Nelson, Tasman, New Zealand

Lakeland Clinical Trials Waikato ( Site 2302)
Nawton, Waikato, New Zealand

Lakeland Clinical Trials Wellington ( Site 2303)
Upper Hutt, Wellington, New Zealand

Pacific Clinical Research Network West Auckland ( Site 2301)
Auckland, New Zealand

Optimal Clinical Trials North ( Site 2308)
Auckland, New Zealand

Optimal Clinical Trials ( Site 2306)
Auckland, New Zealand

Przychodnia EuroMediCare, Wroclaw Lowiecka ( Site 2611)
Wrocław, Dolnoslaskie, Poland

NZOZ GynCentrum - Oddział Kraków ( Site 2609)
Krakow, Malopolskie, Poland

NZOZ GynCentrum - Oddział Bielsko-Biała ( Site 2602)
Bielsko-Biała, Slaskie, Poland

Clinical Medical Research ( Site 2604)
Katowice, Slaskie, Poland

Holsamed ( Site 2603)
Katowice, Slaskie, Poland

PL Certus ( Site 2613)
Poznan, Wielkopolskie, Poland

Investigadores del Este LLC ( Site 4001)
Humacao, Puerto Rico

Miralles Clinical Research LLC ( Site 4004)
San Juan, Puerto Rico

MV HEALTH SERVICES LLC ( Site 4003)
San Juan, Puerto Rico

Spitalul Clinic de Boli Infecțioase și Tropicale Victor Babeș ( Site 2701)
București, Bucuresti, Romania

Centrul Medical SANA ( Site 2704)
Bucuresti, Romania

Spitalul Clinic de Boli Infecțioase ( Site 2703)
Cluj, Romania

Spitalul Clinic de Boli Infecțioase ( Site 2702)
Constanta, Romania

Hospital General Universitario de Elche-Infectius Disease ( Site 3105)
Elche, Alicante, Spain

Hospital Germans Trias i Pujol ( Site 3101)
Badalona, Barcelona, Spain

EAP Osona Sud - Alt Congost S.L.P ( Site 3107)
Centelles, Barcelona, Spain

Hospital Universitari Vall d'Hebron ( Site 3102)
Barcelona, Cataluna, Spain

Hospital Santa Lucia-Medicina Infecciosas ( Site 3106)
Cartagena, Murcia, Spain

EAP Sardenya ( Site 3109)
Barcelona, Spain

Kaohsiung Medical University Chung-Ho Memorial Hospital ( Site 3306)
Kaoshiung, Kaohsiung, Taiwan

Taoyuan General Hospital ( Site 3300)
Taoyuan City, Taoyuan, Taiwan

Kaohsiung Veterans General Hospital ( Site 3307)
Kaohsiung, Taiwan

Taichung Veterans General Hospital ( Site 3305)
Taichung, Taiwan

National Taiwan University Hospital ( Site 3301)
Taipei, Taiwan

Tri-Service General Hospital ( Site 3304)
Taipei, Taiwan

EUROMEDCLINIC ( Site 3517)
Cherkasy, Cherkaska Oblast, Ukraine

MUNICIPAL NON-PROFIT ENTERPRISE CENTRAL CITY CLINICAL HOSPITAL OF CHERNIVTSI CITY COUNCIL ( Site 351
Chernivtsi, Chernihivska Oblast, Ukraine

Clinical medical and diagnostic center Limited Liability Company "Simedgroup" ( Site 3524)
Ivano-Frankivsk, Ivano-Frankivska Oblast, Ukraine

Regional Phthisiology and Pulmonology Center ( Site 3523)
Ivano-Frankivsk, Ivano-Frankivska Oblast, Ukraine

Private Enterprise Private Manufacturing Company Acinus-Medical and Diagnostic Centre ( Site 3537)
Kropyvnytskyi, Kirovohradska Oblast, Ukraine

Medical Center "Harmoniya Krasy" ( Site 3545)
Kyiv, Kyivska Oblast, Ukraine

Edelweiss Medics ( Site 3503)
Kyiv, Kyivska Oblast, Ukraine

Communal Non-Profit Enterprise "Kyiv City Clinical Hospital #1"-Department of Clinical Research ( Si
Kyiv, Kyivska Oblast, Ukraine

Medbud Clinic-Treatment prevention unit ( Site 3506)
Kyiv, Kyivska Oblast, Ukraine

Medical Center of Limited ( Site 3546)
Kyiv, Kyivska Oblast, Ukraine

Center of Family Medicine Plus ( Site 3502)
Kyiv, Kyivska Oblast, Ukraine

Polyclinic of Communal 4th city clinical hospital ( Site 3501)
Lviv, Lvivska Oblast, Ukraine

Municipal non-profit enterprise "Lviv Territorial Medical Union "Multidisciplinary Clinical Hospital
Lviv, Lvivska Oblast, Ukraine

Municipal Enterprise "Volyn Regional Clinical Hospital" of Volyn Regional Council ( Site 3530)
Lutsk, Volynska Oblast, Ukraine

Medlight Clinic ( Site 3548)
Kyiv, Ukraine

Kyiv Railway Clinical Hospital No.2 of Branch Health Center -Center of Clinical Trials ( Site 3549)
Kyiv, Ukraine

Royal Victoria Infirmary ( Site 3608)
Newcastle, Newcastle Upon Tyne, United Kingdom

Lakeside Surgery ( Site 3600)
Northamptonshire, United Kingdom

Contacts

Toll Free Number
1-888-577-8839
Trialsites@msd.com

Medical Director, Study Director
Merck Sharp & Dohme LLC

Merck Sharp & Dohme LLC
NCT Number
MeSH Terms
COVID-19
Coronavirus Infections
Molnupiravir