Official Title
A Phase 1, Randomized, Double-Blinded, Placebo-Controlled, First-in-Human Study to Evaluate the Safety, Tolerability, and Pharmacokinetics of Single-Ascending and Multiple-Ascending Doses of Oral CDI-988 in Healthy Adult Participants
Brief Summary

The goal of this clinical trial is to learn about the safety and pharmacokinetics (PK,the amount of drug in the blood) of a new drug called CDI-988 in healthy volunteers.The main questions it aims to answer are: - Are there any side effects of the drug? - What is the amount of drug that reaches the bloodstream? Participants will be assigned by chance to take either CDI-988 or placebo by mouth and have physical exams, electrocardiograms (ECGs), vital signs, and blood tests to look for any side effects.

Detailed Description

CDI-988 is a severe acute respiratory syndrome coronavirus-2 (SARS-CoV-2)
3-chymotrypsin-like (3CL) protease inhibitor for oral administration. This study is being
conducted in 2 parts to examine the safety, tolerability, and PK of CDI-988 in healthy
participants. Part 1 will entail escalating single doses in sequential cohorts and Part 2
will enroll escalating multiple-dose cohorts. Participants will be monitored for adverse
events, vital signs, laboratory values, and electrocardiograms (ECGs).

Recruiting
Healthy Volunteers

Drug: CDI-988

SARS-CoV-2 3CL protease inhibitor

Drug: Placebo

matching placebo

Eligibility Criteria

Inclusion Criteria:

- Healthy males or non-pregnant, non-lactating females

- Body weight of at least 45 kg.

- Body mass index ≥18.0 and ≤32.0 kg/m2

- Good state of mental and physical health

- Negative severe acute respiratory syndrome coronavirus 2 (SARS-CoV-2) test

Exclusion Criteria:

- Received an investigational drug within 30 days

- Received a coronavirus disease 2019 (COVID-19) vaccine within 7 days

- Drug or alcohol abuse in the past 12 months

- Clinically significant abnormal biochemistry, hematology, coagulation, urinalysis
test results

- Clinically significant abnormal ECG or vital signs

Eligibility Gender
All
Eligibility Age
Minimum: 18 Years ~ Maximum: 55 Years
Countries
Australia
Locations

Scientia Clinical Research Pty Ltd
Randwick, New South Wales, Australia

Contacts

Sam Lee, PhD
425-750-7208
slee@cocrystalpharma.com

Christopher Argent, MD, Principal Investigator
Scientia Clinical Research

Cocrystal Pharma, Inc.
NCT Number
Keywords
Coronavirus
SARS-CoV-2